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65

抑制剂 & 化合物

10

天然产物

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Cat. No. Product Name Target Signaling Pathways
T8310 MMP-9-IN-1

MMP Proteases/Proteasome
MMP-9-IN-1 是特异性的基质金属蛋白酶-9 抑制剂,选择性靶向 MMP-9 的血红素域,对其他 MMP 无影响。
T10425 AZ084

CCR Immunology/Inflammation; Microbiology/Virology
AZ084 是可口服的选择性 CCR8变构拮抗剂,其Ki 值为 0.9 nM,可研究哮喘。
T5465 PF-5274857

PF-5274857 freebase

Smo Stem Cells
PF-5274857 (PF-5274857 free base) freebase 是有效的、具有口服活性的、选择性的、可透过血脑屏障的 Smo 拮抗剂,其 IC50=5.8 nM,Ki=4.6 nM。它有用于包括激活的 Hh 途径驱动的脑肿瘤和脑转移在内的多种肿瘤的研究潜力。
T36758 CAIX Inhibitor S4

S4

Carbonic Anhydrase Metabolism
CAIX Inhibitor S4 (S4) 是一种有效的碳酸酐酶 IX/XII 抑制剂,Ki 分别为 7 nM 和 2 nM。 CA II 和 CA I 的 Ki 分别为 546 和 5600 nM。
T24642 YH-306

YH306,TRV055 acetate (25849-90-5 Free base)

MMP; MMP; FAK; Rho; PI3K; Src Angiogenesis; Cell Cycle/Checkpoint; Cytoskeletal Signaling; PI3K/Akt/mTOR signaling; Proteases/Proteasome; Tyrosine Kinase/Adaptors
YH-306 (TRV055 acetate ) 是 FAK 信号通路的调节剂。 YH-306 显示出抗肿瘤活性,抑制结直肠肿瘤的生长和转移。
T9963 MPT0B390

HDAC Chromatin/Epigenetic; DNA Damage/DNA Repair
MPT0B390 是 HDAC 抑制剂和 TIMP3 诱导剂,可抑制肿瘤生长、转移和血管生成。
T28212 NSC668394

NSC-668394,NSC 668394

PKC Chromatin/Epigenetic; Cytoskeletal Signaling
NSC668394 是一种有效的小分子 ezrin (Thr567) 磷酸化抑制剂。NSC668394 具有潜在的抗肿瘤活性,抑制 ezrin T567 磷酸化,增加 Ca2+依赖性ezrin裂解。NSC668394 可用于研究肿瘤转移。
T27613 inS3-54-A26

STAT JAK/STAT signaling; Stem Cells
inS3-54-A26 是 STAT3 的 DNA 结合域的抑制剂。 inS3-54-A26 抑制肿瘤生长、转移和 STAT3 的基因表达。
T15574 Incyclinide

COL-3,CMT-3

MMP Proteases/Proteasome
Incyclinide (COL-3) 是一种基质金属蛋白酶 (MMP) 抑制剂,能够诱导细胞外基质降解,抑制血管生成,肿瘤生长和侵袭以及转移。
T9107 NP-G2-044

Others Others
NP-G2-044 是fascin 蛋白抑制剂,具有口服活性,IC50值约为 2 μM。它可阻断肿瘤转移并增强抗肿瘤免疫应答。
T6011 Batimastat

巴马司他,BB94

MMP Proteases/Proteasome
Batimastat (BB94) 是广谱MMP 抑制剂,能够抑制MMP-1 (IC50:3 nM),MMP-2 (IC50:4 nM),MMP-9 (IC50:4 nM),MMP-7 (IC50:6 nM) 和 MMP-3 (IC50:20 nM)。
TP1472 Tyroserleutide

Others Others
Tyroserleutide 是一种可从猪脾脏的降解产物中分离得到的小分子三肽,在体内外均对肿瘤生长具有抑制作用。
T14496 BAMB-4

ITPKA-IN-C14

Others Others
BAMB-4 (ITPKA-IN-C14) 是一种新型的膜渗透型ITPKA 抑制剂,在ADP-Glo 实验中的IC50值为37uM。
T26629 Angstrom6

A-6,A 6 peptide,A6,A 6,A6 peptide,A-6 peptide

PAI-1 Metabolism
Angstrom6 (A-6 peptide) 是一种从单链尿激酶纤溶酶原激活剂(scuPA)中提取的 8 肽,它能干扰 uPA/uPAR 级联反应并抑制下游效应。Angstrom6 具有抗肿瘤活性,能通过与 CD44 结合并调节 CD44 介导的细胞信号传导,抑制肿瘤细胞的迁移、侵袭和转移。
T77059 Leronlimab

PRO 140

CCR Immunology/Inflammation; Microbiology/Virology
Leronlimab (PRO 140) 是一种人源化 IgG4 抗 CCR5 单克隆抗体。leronlimumab 具有抗 HIV 病毒活性和抗肿瘤活性, 抑制 CCR 介导的 HIV-1 病毒和小鼠肿瘤模型中癌细胞转移。Leronlimab 可用于研究 HIV 非酒精性脂肪性肝炎 (NASH) 和乳腺癌。
T9398 NSC 73150

NSC 97967

Others Others
6-methyl-2-[2-[(E)-(6-oxo-1-cyclohexa-2,4-dienylidene)methyl]hydraziny l]-1H-pyrimidin-4-one (NSC 73150) 是一种嘧啶衍生物,具有抗肿瘤活性,临床前研究表明,它可以抑制各种肿瘤细胞系的生长,包括乳腺癌、肺癌和肝癌,也被发现可诱导细胞凋亡、抑制血管生成和抑制肿瘤转移。
T29231 ZLD1039

ZLD-1039,ZLD 1039

Histone Methyltransferase Chromatin/Epigenetic
ZLD1039 是一种口服有效的、高选择性 EZH2 抑制剂。ZLD1039 高效抑制 EZH2 野生型及 Y641F 和 A677G 突变型,IC50 分别为 5.6、15 和 4.0 nM。ZLD1039 抑制乳腺肿瘤的生长和转移。
TP1526L1 Fibronectin CS1 Peptide acetate

Others Others
Fibronectin CS1 Peptide acetate 存在于 III 型同源连接段 (IIICS) 以及 C-274(细胞结合结构域)中。 Fibronectin CS1 Peptide 缺乏含有 Arg-Gly-Asp 的结构域,在自发和实验性转移模型中积极抑制肿瘤转移。
TP1345 Kisspeptin-10, human (TFA)(374675-21-5,FREE)

GPR; Kisspeptin Endocrinology/Hormones; GPCR/G Protein
Kisspeptin-10, human (TFA)(374675-21-5,FREE) 是一种有效的血管收缩剂和血管生成抑制剂。 Kisspeptin-10,人类 TFA 通过其受体 GPR54 充当肿瘤转移抑制因子。 Kisspeptin-10-GPR54系统在胚胎肾发育中发挥重要作用。 Kisspeptin-10/GPR54 信号通过 NFATc4 介导的 BMP2 表达诱导成骨细胞分化
T77743 TT-012

Others Others
TT-012 具有抗肿瘤活性,选择性结合动态 MITF,并破坏后者的二聚体形成和 DNA 结合。TT-012 对 B16F10 黑色素瘤细胞中 MITF 的转录有抑制作用。TT-012 在动物模型中对 MITF黑色素瘤细胞的生长和肿瘤生长转移有抑制作用。TT-012 对肝脏和免疫细胞具有较少的细胞毒性。
T25765 LY52

LY-52,LY 52

LY52 is a matrix metalloproteinase-2 inhibitor. It acts by suppressing tumor invasion and metastasis.
T24954 YF479

YF-479,YF 479

YF479 is an inhibitor of histone deacetylase that acts by inhibiting breast tumor growth, metastasis, and recurrence.
T13961 Vitamin CK3

维生素CK3

Others Others
Vitamin CK3 is the combination of Vitamin C and vitamin K3 and has been shown to inhibit tumor growth and lung metastasis.
T69503 ABT-518

ABT-518 is an inhibitor of matrix metalloproteinases, which are associated with tumor growth and development of metastasis.
T71351 STAT3-IN-A69

STAT3-IN-A69 is an inhibitor targeting the DNA-binding domain of STAT3, suppressing tumor growth, metastasis and STAT3 target gene expression in vivo.
T28478 PZ-285

PZ 285

PZ-285 is a potent anticancer agent with similar antitumor activity to the clinically active agent Dox. Pz 285 improves survival, inhibits primary tumor regrowth, and inhibits lung tumor metastasis compared to vehicle control animals.
T70051 MMI-166

MMI-166 is a selective matrix metalloproteinase (MMP) inhibitor that prevents tumor invasion and metastasis by downregulating the activity of MMP-2 and MMP-9.
T70052 S-3304

S-3304 is a n orally-agent agent with potential antineoplastic activity. S-3304 inhibits matrix metalloproteinases (MMPs), thereby inducing extracellular matrix degradation, and inhibiting angiogenesis, tumor growth and invasion, and metastasis.
T61118 CD73-IN-12

CD73-IN-12 is a highly effective CD73 inhibitor that displays strong potential in tumor suppression. CD73, an enzyme intricately linked to tumor development, angiogenesis, and metastasis, is significantly inhibited by CD73-IN-12. This compound holds promise in the formulation of therapeutic medications targeting tumor-related diseases[1].
T10273 AhR modulator-1

Others Others
AhR modulator-1 is a selective and orally active aryl hydrocarbon receptor (AhR) modulator. It inhibits metastasis, in part, by inhibiting prostatic VEGF production prior to tumor formation. It also possesses anti-estrogenic properties in rat uterus.
T35495 (±)13(14)-DiHDPA

(±)13(14)-DiHDPA is a metabolite of docosahexaenoic acid that is produced via oxidation by cytochrome P450 epoxygenases. Epoxygenase metabolites of DHA, including (±)13(14)-DiHDPA, are reported to inhibit angiogenesis, tumor growth, and metastasis.
T22343 HKB99

Others Others
HKB99, an allosteric inhibitor of phosphoglycerate mutase 1, could suppresse tumor growth and metastasis and overcome erlotinib resistance in non-small-cell lung cancer (NSCLC)
T61090 CD73-IN-8

CD73-IN-8, a potent CD73 inhibitor, prevents the catalytic activity of CD73, an enzyme responsible for converting extracellular 5'-phosphate adenosine (5'-AMP) to adenosine. Adenosine, once produced, can induce immunosuppressive effects and facilitate tumor proliferation and/or metastasis. Therefore, CD73-IN-8 holds promise in the development of therapeutic interventions for tumor-related diseases[1].
T80992 Thrombospondin (TSP-1)-derived CD36 binding motif

Thrombospondin (TSP-1)-derived CD36 binding motif 是一种源自基质结合糖蛋白TSP-1的生物活性肽,具备与CD36相互作用的关键结合基序。该肽通过二硫键形成环状结构,与癌症转移、肿瘤粘附和新血管形成等过程相关。研究表明,它能竞争性抑制血小板聚集和肿瘤转移。
T81708 Nagrestipen

Nagrestipen 是一种人巨噬细胞炎症蛋白-1α 变体,也称为 ECI 301,主要用于癌症、肿瘤、转移、放射肿瘤学以及肿瘤转移研究试验,具有显著的抗肿瘤活性。
T69028 CJ-463

CJ-463 is a potent ans selective uPA inhibitor. Treatment with CJ-463 resulted in a significant inhibition of primary tumor growth, with the highest efficacy seen in the 100 mg/kg group. Urokinase (uPA) plays a crucial role in carcinogenesis by facilitating tumor cell invasion and metastasis. CJ-463 may be a novel agent for treatment of lung cancer.
T82645 Cyclic PSAP peptide

Cyclic PSAP peptide(DWLPK)是一种环五肽,具有活性分子特性,在体内能够抑制肿瘤转移扩散和发展。
T71187 Foretinib phosphate

Foretinib phosphate is an orally bioavailable small molecule with potential antineoplastic activity. MET/VEGFR2 inhibitor GSK1363089 binds to and selectively inhibits hepatocyte growth factor (HGF) receptor c-MET and vascular endothelial growth factor receptor 2 (VEGFR2), which may result in the inhibition of tumor angiogenesis, tumor cell proliferation and metastasis. The proto-oncogene c-MET has been found to be over-expressed in a variety of cancers.
T60779 CD73-IN-13

CD73-IN-13 可用于制备肿瘤相关疾病的药物。CD73-IN-13 是CD73的有效抑制剂,CD73 与肿瘤生长、血管生成和转移密切相关。
TP1526 Fibronectin CS1 Peptide

he connecting segment 1 (CS-1) is a cell attachment domain located in the type III homology connecting segment (IIICS) of fibronectin. CS1 peptide of fibronectin, which lacks the Arg-Gly-Asp-containing domain, actively inhibits tumor metastases in spontan
T78826 LN5P45

LN5P45为一种OTUB2抑制剂(IC50: 2.3 μM),能诱导OTUB2在赖氨酸31位点发生单泛素化,适用于探究肿瘤进展与转移。
T70344 BJ-2302

BJ-2302 is a SRC inhibitor. BJ-2302 effectively suppressed MDA-MB-231 cell invasion (Matrigel invasion assay) and metastasis (chorioallantoic membrane assay xenografted with MDA-MB-231-luc2-tdTomato cancer cells). Additionally, BJ-2302 (1 mg/kg) strongly suppressed TNBC cell proliferation in vitro and tumor growth in a xenograft mouse tumor model. The anti-metastatic and anti-tumor effects of BJ-2302 were superior to those of Z-FL-COCHO (1 mg/kg) or batimastat (30 mg/kg), a pan-MMP inhibitor.
T79284 IR-251

IR-251是一种线粒体靶向的近红外荧光探针,通过OATP导向线粒体,诱导肿瘤细胞中线粒体损伤。IR-251抑制PPARγ,从而引发ROS的过量生成,进而抑制β-catenin信号通路及相关细胞周期和转移的下游蛋白,有效抑止肿瘤的增殖和转移。
T75154 ATU027

ATU027, 一种可沉默血管内皮中PKN3表达的siRNA, 已在小鼠癌症模型中证明能有效抑制局部肿瘤侵袭及淋巴结和肺转移。
T61000 CD73-IN-10

CD73-IN-10 可用于肿瘤相关疾病药物的制备。CD73-IN-10 是 CD73的有效抑制剂, 能够催化细胞外5'-磷酸腺苷 (5'-AMP) 产生腺苷。腺苷具有诱导免疫抑制的作用,能够促进肿瘤增殖和/或转移。
T60844 CD73-IN-9

CD73-IN-9 是 CD73 的有效抑制剂,可用于制备治疗肿瘤相关疾病的药物。CD73 可以催化细胞外5'-磷酸腺苷 (5'-AMP) 产生腺苷。腺苷能够诱导免疫抑制作用,并且促进肿瘤增殖和/或转移。
T60599 CD73-IN-7

CD73-IN-7 是一种有效的CD73抑制剂,可用于制备治疗肿瘤相关疾病的药物。CD73 催化细胞外5'-磷酸腺苷 (5'-AMP) 产生腺苷,从而诱导免疫抑制作用并促进肿瘤增殖和/或转移。
T35587 Ganglioside GD1a mixture (sodium salt)

Ganglioside B1

Ganglioside GD1a is a sialic acid-containing glycosphingolipid found in brain, erythrocytes, bone marrow, testis, spleen, and liver. [1] It can be shed from the surface of tumor cells into the microenvironment where it influences tumor-host cell interactions to promote tumor cell proliferation, invasion, and metastasis. Ganglioside GD1a (20 μM) also increases endothelial cell proliferation. Furthermore, ganglioside GD1a has been shown to act as a functional coreceptor for toll-like receptor 2 (T...
T80127 FITC-Ahx-Gly-Arg-Gly-Asp-Ser-Pro

Integrin Cytoskeletal Signaling
FITC-Ahx-Gly-Arg-Gly-Asp-Ser-Pro为FITC标记的GRGDSP,后者为整联蛋白(integrin)抑制剂,能阻止肿瘤细胞与血管内皮细胞粘附,进而抑制肿瘤转移。
T61053 CD73-IN-11

CD73-IN-11 可用于肿瘤相关疾病的药物制备。CD73-IN-11 是 CD73的有效抑制剂。CD73 可以催化细胞外5'-磷酸腺苷 (5'-AMP) 产生腺苷,从而诱导免疫抑制并促进肿瘤增殖和/或转移。

化合物

MMP-9-IN-1
Cat.No: T8310
Synonym:
Target: MMP
AZ084
Cat.No: T10425
Synonym:
Target: CCR
PF-5274857
Cat.No: T5465
Synonym: PF-5274857 freebase
Target: Smo
CAIX Inhibitor S4
Cat.No: T36758
Synonym: S4
Target: Carbonic Anhydrase
YH-306
Cat.No: T24642
Synonym: YH306,TRV055 acetate (25849-90-5 Free base)
Target: MMP, MMP, FAK, Rho, PI3K, Src
MPT0B390
Cat.No: T9963
Synonym:
Target: HDAC
NSC668394
Cat.No: T28212
Synonym: NSC-668394,NSC 668394
Target: PKC
inS3-54-A26
Cat.No: T27613
Synonym:
Target: STAT
Incyclinide
Cat.No: T15574
Synonym: COL-3,CMT-3
Target: MMP
NP-G2-044
Cat.No: T9107
Synonym:
Target: Others
Batimastat
Cat.No: T6011
Synonym: 巴马司他,BB94
Target: MMP
Tyroserleutide
Cat.No: TP1472
Synonym:
Target: Others
BAMB-4
Cat.No: T14496
Synonym: ITPKA-IN-C14
Target: Others
Angstrom6
Cat.No: T26629
Synonym: A-6,A 6 peptide,A6,A 6,A6 peptide,A-6 peptide
Target: PAI-1
Leronlimab
Cat.No: T77059
Synonym: PRO 140
Target: CCR
NSC 73150
Cat.No: T9398
Synonym: NSC 97967
Target: Others
ZLD1039
Cat.No: T29231
Synonym: ZLD-1039,ZLD 1039
Target: Histone Methyltransferase
Fibronectin CS1 Peptide acetate
Cat.No: TP1526L1
Synonym:
Target: Others
Kisspeptin-10, human (TFA)(374675-21-5,FREE)
Cat.No: TP1345
Synonym:
Target: GPR, Kisspeptin
TT-012
Cat.No: T77743
Synonym:
Target: Others
LY52
Cat.No: T25765
Synonym: LY-52,LY 52
Target:
YF479
Cat.No: T24954
Synonym: YF-479,YF 479
Target:
Vitamin CK3
Cat.No: T13961
Synonym: 维生素CK3
Target: Others
ABT-518
Cat.No: T69503
Synonym:
Target:
STAT3-IN-A69
Cat.No: T71351
Synonym:
Target:
PZ-285
Cat.No: T28478
Synonym: PZ 285
Target:
MMI-166
Cat.No: T70051
Synonym:
Target:
S-3304
Cat.No: T70052
Synonym:
Target:
CD73-IN-12
Cat.No: T61118
Synonym:
Target:
AhR modulator-1
Cat.No: T10273
Synonym:
Target: Others
(±)13(14)-DiHDPA
Cat.No: T35495
Synonym:
Target:
HKB99
Cat.No: T22343
Synonym:
Target: Others
CD73-IN-8
Cat.No: T61090
Synonym:
Target:
Thrombospondin (TSP-1)-derived CD36 binding motif
Cat.No: T80992
Synonym:
Target:
Nagrestipen
Cat.No: T81708
Synonym:
Target:
CJ-463
Cat.No: T69028
Synonym:
Target:
Cyclic PSAP peptide
Cat.No: T82645
Synonym:
Target:
Foretinib phosphate
Cat.No: T71187
Synonym:
Target:
CD73-IN-13
Cat.No: T60779
Synonym:
Target:
Fibronectin CS1 Peptide
Cat.No: TP1526
Synonym:
Target:
LN5P45
Cat.No: T78826
Synonym:
Target:
BJ-2302
Cat.No: T70344
Synonym:
Target:
IR-251
Cat.No: T79284
Synonym:
Target:
ATU027
Cat.No: T75154
Synonym:
Target:
CD73-IN-10
Cat.No: T61000
Synonym:
Target:
CD73-IN-9
Cat.No: T60844
Synonym:
Target:
CD73-IN-7
Cat.No: T60599
Synonym:
Target:
Ganglioside GD1a mixture (sodium salt)
Cat.No: T35587
Synonym: Ganglioside B1
Target:
FITC-Ahx-Gly-Arg-Gly-Asp-Ser-Pro
Cat.No: T80127
Synonym:
Target: Integrin
CD73-IN-11
Cat.No: T61053
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T1181 Gefitinib

ZD1839,吉非替尼

EGFR; Tyrosine Kinases; Autophagy Angiogenesis; Autophagy; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Gefitinib (ZD1839) 是一种 EGFR 一代抑制剂,具有口服活性,抑制 EGFR 19 Del 和 L858R 突变。Gefitinib 具有抗肿瘤活性,用于治疗 EGFR 突变的非小细胞肺癌。Gefitinib 用药会产生 EGFR C797S 耐药突变。
T2982 Xanthone

Genicide,呫吨酮,氧杂蒽酮,Xanthenone,Benzophenone oxide

Apoptosis; Others; Influenza Virus; Antibacterial; Antifungal Apoptosis; Microbiology/Virology; Others
Xanthone (Xanthenone) 是一种从山竹果中分离得到的天然产物,具有抗炎,抗氧化,抗肿瘤,抗过敏,抗细菌,抗真菌和抗病毒活性。在癌变的不同阶段可控制细胞分裂和生长,凋亡,炎症和转移。
T8169 Decursinol

Others Others
Decursinol 是一种分离自Angelica gigas 的根中的、口服具有活性的抗伤害药物。它具有抗肿瘤和抗转移作用。
T3402 20(S)-Ginsenoside Rg3

20(S)-人参皂苷 Rg3,人参皂苷 Rg3,20(S)-Ginsenoside-Rg3,Rg3,20S-Ginsenoside Rg3,Ginsenoside Rg3,S-Ginsenoside Rg3

EGFR; Beta Amyloid; Potassium Channel; NF-κB; COX; Sodium Channel; Endogenous Metabolite Angiogenesis; Immunology/Inflammation; JAK/STAT signaling; Membrane transporter/Ion channel; Metabolism; Neuroscience; NF-κB; Tyrosine Kinase/Adaptors
20(S)-Ginsenoside Rg3 (Rg3) 是红参的主要成分,通过抑制肿瘤细胞的粘附和侵袭来抑制肿瘤细胞肺转移。它抑制Na+和hKv1.4通道,IC50分别为 32.2±4.5 和 32.6±2.2 μM。它还抑制Aβ,NF-κB 活性和COX-2表达,抑制人脐静脉内皮细胞的增殖并具有抗血管生成活性。
T75643 Isoxanthohumol

HSV Microbiology/Virology
Isoxanthohumol 是一种从啤酒花和啤酒中提取的一种前黄酮类化合物,对几种人类癌细胞株具有抗增殖活性。Isoxanthohumol对肿瘤细胞肺转移灶的转移或侵袭有抑制作用。Isoxanthohumol具有抗病毒活性,对疱疹病毒(HSV1和HSV2)和牛病毒性腹泻病毒(BVDV)具有抑制作用。
T3229 Cytochalasin D

ATPase; p38 MAPK; Calcium Channel; Akt; PI3K Cytoskeletal Signaling; MAPK; Membrane transporter/Ion channel; Metabolism; PI3K/Akt/mTOR signaling
Cytochalasin D is an actin inhibitor, the removal of actin stress fibers is crucial for the chondrogenic differentiation. It may be an inhibitor of some fertilization processes such as sperm penetration or sperm head decondensation. Cytochalasin D inhibit
T23773 Barbigerone

Barubigeron

Barbigerone is a tumor angiogenesis, growth, and metastasis inhibitor in melanoma.
TN4166 Griffipavixanthone

ERK; Raf; ROS; MEK; Caspase Apoptosis; Immunology/Inflammation; MAPK; Proteases/Proteasome
Griffipavixanthone inhibits the growth of human Non-small-cell lung cancer H520 cells in dose- and time-dependent manners, it induces cell apoptosis through mitochondrial apoptotic pathway accompanying with ROS production. It can inhibit tumor metastasis
TN3587 Capillarisin

MMP; ERK; IL Receptor; BCL; VEGFR; TNF; NOS; NF-κB; TLR; MAPK; COX; DNA/RNA Synthesis; Prostaglandin Receptor; JNK; STAT Angiogenesis; Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair; GPCR/G Protein; Immunology/Inflammation; JAK/STAT signaling; MAPK; Neuroscience; NF-κB; Proteases/Proteasome; Stem Cells; Tyrosine Kinase/Adaptors
Capillarisin is a novel blocker of STAT3 activation and thus may have a potential in negative regulation of growth, metastasis, and chemoresistance of tumor cells, it inhibits cancer cell growth of osteosarcoma cells by inducing apoptosis accompanied with
T35624 Ajoene

Ajoene is a disulfide that has been found inA. sativumand has diverse biological activities, including antibacterial, anticancer, antiplatelet, and antioxidant properties.1,2,3,4It is active against Gram-positive (MICs = 5-160 &#181g/ml) and Gram-negative bacteria (MICs = 136-200 &#181g/ml), as well as yeasts (MICs = 10-20 &#181g/ml).1Ajoene is cytotoxic to mouse melanoma cells (IC50= 18 &#181M), as well as human colon, lung, mammary, and pancreatic cancer cells (IC50s = 7-41 &#181M).2It reduces...

天然产物

Gefitinib
Cat.No: T1181
Synonym: ZD1839,吉非替尼
Target: EGFR, Tyrosine Kinases, Autophagy
Xanthone
Cat.No: T2982
Synonym: Genicide,呫吨酮,氧杂蒽酮,Xanthenone,Benzophenone oxide
Target: Apoptosis, Others, Influenza Virus, Antibacterial, Antifungal
Decursinol
Cat.No: T8169
Synonym:
Target: Others
20(S)-Ginsenoside Rg3
Cat.No: T3402
Synonym: 20(S)-人参皂苷 Rg3,人参皂苷 Rg3,20(S)-Ginsenoside-Rg3,Rg3,20S-Ginsenoside Rg3,Ginsenoside Rg3,S-Ginsenoside Rg3
Target: EGFR, Beta Amyloid, Potassium Channel, NF-κB, COX, Sodium Channel, Endogenous Metabolite
Isoxanthohumol
Cat.No: T75643
Synonym:
Target: HSV
Cytochalasin D
Cat.No: T3229
Synonym:
Target: ATPase, p38 MAPK, Calcium Channel, Akt, PI3K
Barbigerone
Cat.No: T23773
Synonym: Barubigeron
Target:
Griffipavixanthone
Cat.No: TN4166
Synonym:
Target: ERK, Raf, ROS, MEK, Caspase
Capillarisin
Cat.No: TN3587
Synonym:
Target: MMP, ERK, IL Receptor, BCL, VEGFR, TNF, NOS, NF-κB, TLR, MAPK, COX, DNA/RNA Synthesis, Prostaglandin Receptor, JNK, STAT
Ajoene
Cat.No: T35624
Synonym:
Target:
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